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Version October 2024
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Emetic risk of single, oral antineoplastic agents in adults*
Emetic risk of single, oral antineoplastic agents in adults*
Risk level
Agent
Moderate or high (≥30%)
Abemaciclib
Avapritinib
Bosutinib
Cabozantinib
Ceritinib
Crizotinib
Cyclophosphamide
Enasidenib
Fedratinib
Hexamethylmelamine
Imatinib
Lenvatinib
Lomustine
Midostaurin
Niraparib
Procarbazine
Ribociclib
Rucaparib
Selinexor
TAS-102 (trifluridine-tipiracil)
Temozolomide
Vinorelbine
Minimal or low (<30%)
6-Thioguanine
Acalabrutinib
Afatinib
Alectinib
Alpelisib
Axitinib
Bexarotene
Brigatinib
Capecitabine
Chlorambucil
Cobimetinib
Dabrafenib
Dacomitinib
Dasatinib
Duvelisib
Encorafenib
Entrectinib
Erdafitinib
Erlotinib
Estramustine
Etoposide
Everolimus
Fludarabine
Risk level
Agent
Minimal or low (<30%)
(continued)
Gefitinib
Gilteritinib
Glasdegib
Hydroxyurea
Ibrutinib
Idelalisib
Ivosidenib
Ixazomib
Lapatinib
Larotrectinib
Lenalidomide
Lorlatinib
Melphalan
Methotrexate
Neratinib
Nilotinib
Olaparib
Osimertinib
Palbociclib
Panobinostat
Pazopanib
Pexidartinib
Pomalidomide
Ponatinib
Regorafenib
Ruxolitinib
Sonidegib
Sorafenib
Sunitinib
Talazoparib
Tazemetostat
Tegafur-Uracil
Thalidomide
Topotecan
Trametinib
Vandetanib
Vemurafenib
Venetoclax
Vismodegib
Vorinostat
Zanubrutinib
* The classified emetic potential of oral agents is based on a full course of therapy and not a single dose.
Reproduced with permission from: Hesketh PJ, Kris MG, Basch E, et al. Antiemetics: ASCO guideline update. J Clin Oncol 2020; 38:JCO2001296. Copyright © 2020 American Society of Clinical Oncology. All rights reserved.
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